Assay Report Card

Basic Information

ID: ALA5115449

Type: ADME

Description: Inhibition of CYP2C9 in human kidney microsomes assessed as inhibition of 20-HETE formation using 7-methoxy-4-trifluoromethylcoumarin as substrate in presence of arachidonic acid and NADPH by fluorescence assay

Organism: Homo sapiens

Tissue: Kidney

Subcellular Fraction: Microsome

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
206.292.982.98
255.712.012.01