Basic Information
ID: ALA5116079
Type: Binding
Description: Selectivity ratio of Ki for binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrate to Ki for binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant using Mes-DArg-Pro-Arg-AMC as substrate
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5116079
Ratio Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 661.83 | 3.80 | 3.80 |
| 662.86 | 4.40 | 4.40 |
| 673.67 | 4.92 | 4.92 |
| 633.82 | 3.07 | 3.07 |
| 635.79 | 3.26 | 3.26 |
| 664.83 | 3.63 | 3.63 |
| 676.84 | 3.73 | 3.73 |
| 652.79 | 3.25 | 3.25 |
| 670.78 | 3.39 | 3.39 |
| 690.91 | 4.93 | 4.93 |
| 646.82 | 2.90 | 2.90 |
| 634.80 | 3.11 | 3.11 |
| 634.80 | 3.11 | 3.11 |
| 620.78 | 2.59 | 2.59 |
| 648.83 | 3.76 | 3.76 |
| 622.75 | 2.46 | 2.46 |
| 618.80 | 3.92 | 3.92 |
| 650.80 | 3.24 | 3.24 |
| 633.82 | 3.07 | 3.07 |
| 651.79 | 3.62 | 3.62 |
| 652.79 | 3.25 | 3.25 |
| 646.82 | 2.90 | 2.90 |
| 650.80 | 3.20 | 3.20 |