Assay Report Card

Basic Information

ID: ALA5121925

Type: Binding

Description: Inhibition of human Kv1.3 expressed in HEK293 cells assessed as inhibition of tetracyclin induced current at 30 uM at holding potential of -80 mV by patch clamp method relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
329.373.333.33
600.714.174.17
584.714.964.96
540.654.604.60
645.755.865.86
540.654.604.60
584.714.964.96
540.654.604.60
598.694.144.14
600.714.674.67
496.604.384.38
598.694.294.29
556.653.723.72
556.653.723.72
498.624.034.03
618.723.133.13
645.755.865.86
512.603.353.35
598.694.144.14
626.745.535.53
642.744.654.65