Basic Information
ID: ALA5123805
Type: Binding
Description: Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins by microfluidic capillary electrophoresis analysis
Format: BAO_0000357
Organism: Homo sapiens
Target: Histone-lysine N-methyltransferase, H3 lysine-9 specific 3(ALA6032)
Document: ALA5120862
Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins by microfluidic capillary electrophoresis analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5123805
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 509.74 | 5.84 | 5.84 |
| 478.64 | 4.09 | 4.09 |
| 554.74 | 5.75 | 5.75 |
| 492.67 | 4.33 | 4.33 |
| 479.63 | 4.05 | 4.05 |
| 518.71 | 5.01 | 5.01 |
| 554.74 | 5.66 | 5.66 |
| 506.70 | 4.87 | 4.87 |
| 464.61 | 3.70 | 3.70 |
| 528.70 | 5.24 | 5.24 |
| 506.70 | 4.52 | 4.52 |
| 504.68 | 4.62 | 4.62 |
| 492.62 | 3.73 | 3.73 |
| 464.61 | 3.70 | 3.70 |
| 506.70 | 4.87 | 4.87 |
| 492.67 | 4.11 | 4.11 |
| 492.67 | 4.11 | 4.11 |
| 492.67 | 4.48 | 4.48 |
| 550.71 | 6.26 | 6.26 |
| 438.58 | 3.92 | 3.92 |
| 533.72 | 3.77 | 3.77 |
| 474.61 | 4.69 | 4.69 |
| 492.67 | 4.13 | 4.13 |
| 502.66 | 4.09 | 4.09 |
| 402.54 | 2.52 | 2.52 |
| 490.65 | 4.23 | 4.23 |
| 554.74 | 5.66 | 5.66 |
| 528.70 | 5.24 | 5.24 |
| 488.63 | 3.82 | 3.82 |
| 520.68 | 3.86 | 3.86 |
| 388.52 | 2.17 | 2.17 |