Basic Information
ID: ALA5125529
Type: Binding
Description: Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substrate addition and measured after 1 hr by fluorogenic assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK-293T
Target: Histone deacetylase 1(ALA325)
Document: ALA5120930
Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substrate addition and measured after 1 hr by fluorogenic assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5125529
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 415.54 | 3.76 | 3.76 |
| 443.59 | 4.54 | 4.54 |
| 401.51 | 3.71 | 3.71 |
| 325.41 | 2.12 | 2.12 |
| 429.56 | 4.15 | 4.15 |
| 339.44 | 2.68 | 2.68 |
| 401.51 | 3.71 | 3.71 |
| 401.51 | 3.71 | 3.71 |