Basic Information
ID: ALA5125569
Type: Functional
Description: Invivo inhibition of SETD2 in NOD SCID mouse xenografted with human KMS-11 cells assessed as reduction in H3K36me3 at 30 mg/kg, po bid administered starting from day 7 to 37 days post inoculation and measured at 12 hr post last dose
Format: BAO_0000218
Organism: Mus musculus
Target: Unchecked(ALA612545)
Document: ALA5120931
Invivo inhibition of SETD2 in NOD SCID mouse xenografted with human KMS-11 cells assessed as reduction in H3K36me3 at 30 mg/kg, po bid administered starting from day 7 to 37 days post inoculation and measured at 12 hr post last dose: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5125569
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 400.50 | 2.82 | 2.82 |