Assay Report Card

Basic Information

ID: ALA5125630

Type: Binding

Description: PROTAC activity at CBRN/BRD4 in human HEK293T cells assessed as degradation of BRD4 incubated for 24 hrs by HiBiT assay

Organism: Homo sapiens

Cell type: HEK293T

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
115.09-0.48-0.48
785.283.683.68
400.894.274.27
840.363.273.27
345.310.660.66
797.293.783.78
815.313.263.26
876.445.775.77
429.34-0.93-0.93
713.265.365.36
332.27-0.45-0.45
756.334.864.86
731.284.854.85
497.963.803.80
960.474.184.18
248.241.141.14