Basic Information
ID: ALA5125631
Type: Binding
Description: PROTAC activity at CBRN/BRD4 in human HEK293T cells assessed as degradation of BRD4 at 20 mM incubated for 24 hrs by HiBiT assay relative to control
Organism: Homo sapiens
Cell type: HEK293T
Activity Charts
Bioactivity
Activity Types for Assay ALA5125631
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 115.09 | -0.48 | -0.48 |
| 785.28 | 3.68 | 3.68 |
| 400.89 | 4.27 | 4.27 |
| 840.36 | 3.27 | 3.27 |
| 345.31 | 0.66 | 0.66 |
| 797.29 | 3.78 | 3.78 |
| 815.31 | 3.26 | 3.26 |
| 876.44 | 5.77 | 5.77 |
| 429.34 | -0.93 | -0.93 |
| 713.26 | 5.36 | 5.36 |
| 332.27 | -0.45 | -0.45 |
| 756.33 | 4.86 | 4.86 |
| 731.28 | 4.85 | 4.85 |
| 497.96 | 3.80 | 3.80 |
| 960.47 | 4.18 | 4.18 |
| 248.24 | 1.14 | 1.14 |