Basic Information
ID: ALA5125638
Type: Binding
Description: Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substrate measured for 10 mins every 30 seconds by fluorescence microplate reader assay
Organism: Trypanosoma brucei rhodesiense
Activity Charts
Bioactivity
Activity Types for Assay ALA5125638
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 518.06 | 5.64 | 5.64 |
| 469.59 | 4.68 | 4.68 |
| 499.61 | 4.69 | 4.69 |
| 505.57 | 4.96 | 4.96 |
| 487.58 | 4.82 | 4.82 |
| 484.04 | 5.45 | 5.45 |
| 519.65 | 5.84 | 5.84 |
| 449.60 | 4.79 | 4.79 |
| 572.03 | 6.35 | 6.35 |
| 504.03 | 5.34 | 5.34 |
| 483.61 | 4.99 | 4.99 |