Basic Information
ID: ALA5127106
Type: Binding
Description: Agonist activity at 6His-tagged human RORC LBD (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of N-terminal biotinylated SRC1-4 derived QKPTSGPQTPQAQQKSLLQQLLTE coactivator peptide by luminescence based AlphaScreen analysis
Format: BAO_0000219
Organism: Homo sapiens
Target: Nuclear receptor ROR-gamma(ALA1741186)
Document: ALA5126511
Agonist activity at 6His-tagged human RORC LBD (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of N-terminal biotinylated SRC1-4 derived QKPTSGPQTPQAQQKSLLQQLLTE coactivator peptide by luminescence based AlphaScreen analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5127106
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 396.44 | 3.47 | 3.47 |