ID: ALA5127379
Type: Binding
Description: Inhibition of GST-fused human recombinant DYRK1B expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA5127379
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
245.24 | 0.54 | 0.54 |
337.34 | 2.36 | 2.36 |
307.31 | 2.35 | 2.35 |
287.32 | 1.58 | 1.58 |
321.34 | 2.70 | 2.70 |
273.29 | 1.24 | 1.24 |
315.37 | 2.36 | 2.36 |
349.39 | 3.16 | 3.16 |
259.26 | 0.85 | 0.85 |
321.34 | 2.66 | 2.66 |
323.31 | 2.06 | 2.06 |
399.41 | 4.15 | 4.15 |
324.36 | 3.50 | 3.50 |
335.36 | 2.97 | 2.97 |
335.36 | 2.97 | 2.97 |
382.46 | 2.19 | 2.19 |
383.41 | 4.02 | 4.02 |
403.44 | 2.28 | 2.28 |
285.30 | 1.34 | 1.34 |
281.29 | 2.76 | 2.76 |
393.49 | 4.46 | 4.46 |
335.36 | 2.97 | 2.97 |
405.46 | 2.11 | 2.11 |
309.32 | 2.34 | 2.34 |
325.30 | 2.49 | 2.49 |
341.30 | 2.20 | 2.20 |
392.46 | 3.33 | 3.33 |
276.32 | 2.00 | 2.00 |
321.34 | 2.38 | 2.38 |
309.32 | 1.92 | 1.92 |
335.36 | 2.79 | 2.79 |
408.43 | 2.25 | 2.25 |
262.29 | 1.60 | 1.60 |
290.34 | 2.34 | 2.34 |
321.34 | 2.74 | 2.74 |
391.47 | 4.48 | 4.48 |
295.30 | 2.04 | 2.04 |
390.44 | 3.34 | 3.34 |
314.35 | 0.58 | 0.58 |
304.37 | 2.73 | 2.73 |
321.34 | 2.40 | 2.40 |
309.32 | 2.34 | 2.34 |
417.47 | 2.53 | 2.53 |
325.30 | 2.49 | 2.49 |
309.32 | 2.35 | 2.35 |
407.47 | 2.09 | 2.09 |
245.24 | 0.46 | 0.46 |
299.33 | 1.73 | 1.73 |
391.43 | 1.76 | 1.76 |
231.21 | 0.20 | 0.20 |
293.33 | 2.63 | 2.63 |
393.45 | 1.75 | 1.75 |
290.34 | 2.39 | 2.39 |
308.30 | 1.75 | 1.75 |
301.30 | 0.57 | 0.57 |
319.36 | 2.95 | 2.95 |
305.34 | 2.56 | 2.56 |
393.44 | 3.92 | 3.92 |