Basic Information
ID: ALA5128698
Type: Binding
Description: Inhibition of ABCG2 (unknown origin) expressed in human HEK293 cells membrane vesicles assessed inhibition of BCRP- mediated transport of 3[H]-E1S for 1 to 5 mins using [3H]-estrone sulfate as substrate by rapid filtration technique
Organism: Homo sapiens
Cell type: HEK293
Subcellular Fraction: Membrane vesicle
Activity Charts
Bioactivity
Activity Types for Assay ALA5128698
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 378.32 | 4.45 | 4.45 |
| 253.74 | 2.21 | 2.21 |
| 366.84 | 5.51 | 5.51 |