Basic Information
ID: ALA5128959
Type: Binding
Description: Selectivity index, ratio of IC50 for inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) to IC50 for inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 1 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Unchecked(ALA612545)
Document: ALA5126568
Selectivity index, ratio of IC50 for inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) to IC50 for inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 1 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5128959
Ratio IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 362.41 | 3.97 | 3.97 |