Basic Information
ID: ALA5130203
Type: Binding
Description: Antagonist activity at human A2AAR S277A/H278A double mutant expressed in CHO cells assessed as inhibition of CGS21680-induced cAMP accumulation preincubated for 20 mins followed by CGS21680 addition and measured after 20 mins by alpha screen assay
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA5130203
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 399.48 | 1.93 | 1.93 |