Agonist activity at human GLP-1R assessed as increase in ERK1/2 phosphorylation by measuring maximum efficacy at Thr202/Tyr204 residues incubated for ...

Basic Information

ID: ALA5130390

Type: Functional

Description: Agonist activity at human GLP-1R assessed as increase in ERK1/2 phosphorylation by measuring maximum efficacy at Thr202/Tyr204 residues incubated for 20 mins by AlphaLISA assay relative to GLP1

Format: BAO_0000019

Organism: Homo sapiens

Target:  Glucagon-like peptide 1 receptor(ALA1784)

Document:  ALA5126621

Agonist activity at human GLP-1R assessed as increase in ERK1/2 phosphorylation by measuring maximum efficacy at Thr202/Tyr204 residues incubated for 20 mins by AlphaLISA assay relative to GLP1: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
4186.64
3235.66
3251.66
3265.68
4067.52
3353.79
3251.66
3265.68
3281.68
3307.72
3267.66
3235.66
3219.66
4224.73
3281.68
3281.68
3249.68
3251.66
3235.66
3289.79
3265.68