Assay Report Card

Basic Information

ID: ALA5130547

Type: Binding

Description: Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by measuring efficacy at 100 nM measured at 180 sec by fluorescence based microplate reader analysis relative to capsaicin

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
305.423.793.79
372.904.394.39
370.843.363.36
390.373.333.33
390.274.224.22
424.813.983.98
335.413.233.23
351.412.932.93
356.822.972.97
323.361.711.71
356.822.972.97
336.402.622.62
323.361.711.71
390.373.333.33
390.373.333.33
356.822.972.97
336.402.622.62
355.833.573.57
404.304.234.23
401.273.073.07
356.822.972.97
336.402.622.62
404.304.614.61
401.273.073.07
370.842.982.98
352.402.322.32
390.373.333.33
327.433.053.05
336.402.622.62
355.833.573.57
390.274.224.22
352.402.322.32
327.432.952.95
370.842.982.98
390.373.333.33
390.373.333.33
403.315.295.29
356.822.972.97
356.822.972.97
370.843.363.36
335.413.233.23
351.412.932.93
404.304.614.61
424.813.983.98