Basic Information
ID: ALA5133706
Type: Binding
Description: Inhibition of His6-tagged ENL YEATS domain (unknown origin) expressed in Escherichia coli BL21 DE3 and biotinylated H3K27ac peptide interaction using biotin-labeled peptide PRKQLATKAARK(Ac)SAPATGGVKKPH as substrate pretreated for 15 mins followed by substrate addition for 30 mins by AlphaScreen assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Protein ENL(ALA4295801)
Document: ALA5131438
Inhibition of His6-tagged ENL YEATS domain (unknown origin) expressed in Escherichia coli BL21 DE3 and biotinylated H3K27ac peptide interaction using biotin-labeled peptide PRKQLATKAARK(Ac)SAPATGGVKKPH as substrate pretreated for 15 mins followed by substrate addition for 30 mins by AlphaScreen assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5133706
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 388.48 | 3.69 | 3.69 |
| 696.88 | 5.17 | 5.17 |