Basic Information
ID: ALA5134929
Type: Binding
Description: Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins by Fura-2 AM based fluorescence assay
Organism: Homo sapiens
Cell type: 1321N1
Activity Charts
Bioactivity
Activity Types for Assay ALA5134929
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 510.40 | 2.03 | 2.03 |
| 1297.30 | ||
| 407.38 | 4.79 | 4.79 |
| 330.45 | 3.42 | 3.42 |
| 399.34 | 4.73 | 4.73 |
| 393.90 | 4.28 | 4.28 |
| 472.25 | 5.24 | 5.24 |
| 393.53 | 2.36 | 2.36 |
| 758.17 | 4.19 | 4.19 |
| 349.89 | 3.76 | 3.76 |
| 374.51 | 3.73 | 3.73 |
| 461.35 | 5.50 | 5.50 |