Basic Information
ID: ALA5136431
Type: Functional
Description: Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated for 30 mins in presence of GIPR agonist GIP(I-42) by HTRF assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Gastric inhibitory polypeptide receptor(ALA4383)
Document: ALA5131553
Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated for 30 mins in presence of GIPR agonist GIP(I-42) by HTRF assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5136431
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 447.59 | 7.32 | 7.32 |
| 577.61 | 8.08 | 8.08 |