Basic Information
ID: ALA5136938
Type: Binding
Description: Inhibition of recombinant human EHMT2 G9a expressed in Escherichia coli Rosetta2(DE3)pLysS at 100 uM using histone H3 as substrate measured at 120 mins by liquid scintillation counting analysis
Format: BAO_0000019
Organism: Homo sapiens
Target: Histone-lysine N-methyltransferase, H3 lysine-9 specific 3(ALA6032)
Document: ALA5131574
Inhibition of recombinant human EHMT2 G9a expressed in Escherichia coli Rosetta2(DE3)pLysS at 100 uM using histone H3 as substrate measured at 120 mins by liquid scintillation counting analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5136938
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 384.42 | -1.44 | -1.44 |
| 405.42 | -2.24 | -2.24 |
| 381.39 | -2.06 | -2.06 |
| 419.44 | -1.84 | -1.84 |
| 419.44 | -1.85 | -1.85 |
| 433.47 | -1.45 | -1.45 |