Basic Information
ID: ALA5137975
Type: Binding
Description: PROTAC activity at VHL/LSD1/HDAC1/CoREST complex interaction (unknown origin) assessed as induction of HDAC1 degradation using Boc-(Ac)Lys-AMC as substrate incubated for 20 mins by fluorescence based assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Unchecked(ALA612545)
Document: ALA5136981
PROTAC activity at VHL/LSD1/HDAC1/CoREST complex interaction (unknown origin) assessed as induction of HDAC1 degradation using Boc-(Ac)Lys-AMC as substrate incubated for 20 mins by fluorescence based assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5137975
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 852.11 | 7.60 | 7.60 |