Assay Report Card

Basic Information

ID: ALA5140256

Type: Binding

Description: Antagonist activity against human P2X7R stably transfected in human 1321N1 cells assessed as reduction in BzATP-induced activity incubated for 5 to 10 mins by EtBr staining based fluorescence assay

Organism: Homo sapiens

Cell type: 1321N1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1297.30
407.470.910.91
351.393.093.09
316.342.252.25
379.421.191.19
335.772.592.59