Basic Information
ID: ALA5142862
Type: Binding
Description: Inhibition of DNA-PK (unknown origin) using EPPLSQEAFADLWKK peptide as substrate preincubated with compound for 30 mins followed by substrate addition and further incubated for 40 mins in presence of ATP by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5142862
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 380.41 | 1.58 | 1.58 |
| 393.43 | 2.21 | 2.21 |
| 393.46 | 1.49 | 1.49 |
| 393.43 | 2.21 | 2.21 |
| 407.45 | 2.55 | 2.55 |
| 390.45 | 3.08 | 3.08 |
| 391.44 | 2.48 | 2.48 |
| 389.46 | 2.61 | 2.61 |
| 407.45 | 2.55 | 2.55 |
| 391.44 | 2.48 | 2.48 |
| 403.49 | 3.00 | 3.00 |
| 419.49 | 1.97 | 1.97 |
| 389.46 | 2.65 | 2.65 |
| 391.44 | 2.48 | 2.48 |
| 404.48 | 2.39 | 2.39 |
| 431.50 | 2.38 | 2.38 |
| 404.48 | 2.39 | 2.39 |
| 389.46 | 2.61 | 2.61 |
| 433.52 | 2.62 | 2.62 |