Basic Information
ID: ALA5144358
Type: Binding
Description: Inhibition of human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21 (DE3) at 250 nM using KKISGRLSPIMTEQ as substrate incubated in presence of ATP relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5144358
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 411.49 | 3.58 | 3.58 |
| 483.35 | 5.66 | 5.66 |
| 458.42 | 5.32 | 5.32 |
| 418.48 | 5.21 | 5.21 |
| 420.45 | 4.60 | 4.60 |
| 422.44 | 5.04 | 5.04 |
| 429.46 | 4.77 | 4.77 |
| 422.44 | 5.04 | 5.04 |
| 458.50 | 4.59 | 4.59 |
| 418.48 | 4.83 | 4.83 |
| 368.42 | 3.99 | 3.99 |
| 382.45 | 4.38 | 4.38 |
| 438.90 | 5.55 | 5.55 |
| 404.45 | 4.90 | 4.90 |
| 342.38 | 3.60 | 3.60 |
| 472.45 | 5.92 | 5.92 |
| 410.50 | 5.16 | 5.16 |
| 440.51 | 4.45 | 4.45 |
| 422.44 | 5.04 | 5.04 |
| 458.50 | 4.59 | 4.59 |
| 458.42 | 5.32 | 5.32 |
| 429.46 | 4.77 | 4.77 |
| 438.90 | 5.55 | 5.55 |
| 476.49 | 4.72 | 4.72 |
| 440.43 | 5.18 | 5.18 |
| 473.34 | 6.21 | 6.21 |
| 458.50 | 4.59 | 4.59 |