Assay Report Card

Basic Information

ID: ALA5144378

Type: Binding

Description: Binding affinity to C-terminal HiBiT-tagged human DYRK1A (28 to 499 residues) stably expressed in HEK293 cells assessed as thermal stability by measuring increase in DYRK1A in soluble fraction at 10 to 30 uM incubated for 3.5 mins by ITDRF-CETSA analysis

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
418.484.834.83