Assay Report Card

Basic Information

ID: ALA5148371

Type: Binding

Description: Selectivity index, ratio of Ki for displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane to Ki for displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT1R expressed in HEK293 cell membrane

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
547.727.047.04
573.767.587.58