Basic Information
ID: ALA5148527
Type: Binding
Description: Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H]DPCPX addition and measured after 1.5 hrs by TopCount scintillation counting method
Organism: Homo sapiens
Cell type: HEK293
Subcellular Fraction: Membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA5148527
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 315.74 | 3.28 | 3.28 |
| 318.34 | 1.79 | 1.79 |
| 391.26 | 1.79 | 1.79 |