Basic Information
ID: ALA5149651
Type: Binding
Description: Inhibition of full-length N-terminal His-TEV-tagged inactive form of MSK1 (2 to 802 residues) (unknown origin) expressed in HEK293 cells assessed as steady state velocity at 20 times IC50 using ATXN1 peptide as substrate preincubated for 3 hrs followed by dilution with buffer and subsequent addition of substrate and ATP measured up to 7 hrs by jump dilution method (Rvb = 4.76 x 10^-3 No_unit)
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5149651
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 196.21 | 1.82 | 1.82 |
| 230.66 | 2.47 | 2.47 |
| 266.09 | 2.52 | 2.52 |
| 265.10 | 3.33 | 3.33 |