Assay Report Card

Basic Information

ID: ALA5149660

Type: Binding

Description: Covalent binding affinity to N-terminal His-Smt-tagged MSK1 C-terminal kinase domain (414 to 738 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) at 1:1 ratio of enzyme to compound measured after 1 min by LC-MS analysis relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
289.302.022.02
450.503.053.05
230.662.472.47
265.103.123.12
231.651.861.86