Basic Information
ID: ALA5151459
Type: Binding
Description: Displacement of [3H]-histamine from human histamine H4 receptor stably expressed in baculovirus infected Sf9 cell membrane co-expressing G-alphai2 and G-beta1gamma2 incubated for 60 mins by scintillation counting analysis
Organism: Homo sapiens
Cell type: Sf9
Subcellular Fraction: Membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA5151459
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 111.15 | -0.09 | -0.09 |
| 211.33 | 1.58 | 1.58 |
| 600.54 | 3.47 | 3.47 |
| 1118.94 | 4.85 | 4.85 |
| 1052.88 | 0.69 | 0.69 |
| 608.52 | 3.34 | 3.34 |
| 1118.94 | 4.85 | 4.85 |
| 664.63 | 4.32 | 4.32 |
| 446.46 | 1.59 | 1.59 |
| 1024.83 | -0.09 | -0.09 |
| 712.59 | 0.97 | 0.97 |
| 560.48 | 1.47 | 1.47 |
| 678.66 | 4.80 | 4.80 |
| 617.57 | 1.85 | 1.85 |
| 592.54 | 2.33 | 2.33 |
| 540.49 | 1.46 | 1.46 |
| 586.52 | 1.64 | 1.64 |
| 438.36 | 1.57 | 1.57 |
| 539.43 | 0.78 | 0.78 |
| 426.46 | 1.58 | 1.58 |
| 714.54 | 1.10 | 1.10 |
| 597.58 | 1.69 | 1.69 |
| 678.66 | 4.80 | 4.80 |
| 656.65 | 3.10 | 3.10 |
| 558.44 | 1.31 | 1.31 |
| 631.60 | 2.33 | 2.33 |
| 601.51 | 1.39 | 1.39 |
| 555.50 | 1.25 | 1.25 |
| 388.30 | 1.11 | 1.11 |
| 616.59 | 2.46 | 2.46 |
| 595.57 | 1.88 | 1.88 |
| 588.53 | 3.33 | 3.33 |
| 642.62 | 4.35 | 4.35 |
| 561.47 | 0.87 | 0.87 |
| 566.53 | 1.63 | 1.63 |
| 541.48 | 0.86 | 0.86 |
| 642.62 | 2.63 | 2.63 |
| 664.63 | 4.32 | 4.32 |
| 542.44 | 1.72 | 1.72 |
| 420.37 | 1.43 | 1.43 |
| 608.52 | 3.34 | 3.34 |
| 588.53 | 3.33 | 3.33 |
| 480.56 | 2.61 | 2.61 |