Assay Report Card

Basic Information

ID: ALA5151472

Type: Functional

Description: Agonist activity at human histamine H2 receptor stably expressed in HEK293T cells co-expressing ARRB2 assessed as maximum efficacy at 100 uM incubated for 60 mins by beta-arrestin2 recruitment assay relative to histamine

Organism: Homo sapiens

Cell type: HEK293T

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
111.15-0.09-0.09
1024.83-0.09-0.09
560.481.471.47
617.571.851.85
540.491.461.46
438.361.571.57
631.602.332.33
555.501.251.25
388.301.111.11
616.592.462.46
595.571.881.88
561.470.870.87
541.480.860.86
420.371.431.43