Basic Information
ID: ALA5151702
Type: Binding
Description: Inhibition of human 20S proteasome beta5 subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured after 1 hr by fluorescence intensity assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5151702
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 384.25 | ||
| 719.92 | 2.58 | 2.58 |
| 324.15 | ||
| 553.16 | ||
| 364.21 | ||
| 313.12 | ||
| 325.13 | ||
| 277.09 | ||
| 323.16 | ||
| 329.16 | ||
| 350.18 | ||
| 329.16 | ||
| 311.19 | ||
| 247.06 | ||
| 303.12 | ||
| 311.19 | ||
| 329.16 | ||
| 353.18 | ||
| 348.17 | ||
| 249.12 | ||
| 317.58 | ||
| 329.16 | ||
| 446.32 | ||
| 325.13 | ||
| 357.60 | ||
| 291.11 | ||
| 359.62 | ||
| 339.20 | ||
| 324.15 | ||
| 297.16 | ||
| 371.63 | ||
| 337.18 | ||
| 341.15 | ||
| 323.16 | ||
| 303.12 | ||
| 303.12 | ||
| 303.12 | ||
| 384.63 | ||
| 311.19 | ||
| 359.62 | ||
| 283.14 | ||
| 357.60 |