Assay Report Card

Basic Information

ID: ALA5152651

Type: Binding

Description: Inhibition of full length N-terminal GST-tagged human BTK expressed in Sf21 cells assessed as inhibition constant using NH2-KKKAPFSWYLPEEG as substrate in presence of ATP measured for 2 hrs by microplate reader assay

Organism: Homo sapiens

Cell type: Sf21

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
539.625.605.60
520.624.384.38
540.615.075.07
554.635.385.38
478.583.913.91
554.635.385.38
540.615.075.07
532.634.524.52
518.644.794.79
504.624.404.40
520.664.424.42
539.625.685.68
546.654.914.91