Basic Information
ID: ALA5152652
Type: Binding
Description: Inhibition of full length N-terminal GST-tagged human BTK expressed in Sf21 cells assessed as ratio of Kinact/Ki using NH2-KKKAPFSWYLPEEG as substrate in presence of ATP measured for 2 hrs by microplate reader assay
Organism: Homo sapiens
Cell type: Sf21
Activity Charts
Bioactivity
Activity Types for Assay ALA5152652
Ratio
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 539.62 | 5.60 | 5.60 |
| 520.62 | 4.38 | 4.38 |
| 540.61 | 5.07 | 5.07 |
| 554.63 | 5.38 | 5.38 |
| 478.58 | 3.91 | 3.91 |
| 554.63 | 5.38 | 5.38 |
| 540.61 | 5.07 | 5.07 |
| 532.63 | 4.52 | 4.52 |
| 518.64 | 4.79 | 4.79 |
| 504.62 | 4.40 | 4.40 |
| 520.66 | 4.42 | 4.42 |
| 539.62 | 5.68 | 5.68 |
| 546.65 | 4.91 | 4.91 |