ID: ALA5154013
Type: Functional
Description: Antagonist activity at CCR5 (unknown origin) expressed in HEK293 cells co-expressing Galpha16 assessed as intracellular calcium change incubated for 15 mins by Fluo-4 AM calcium flux assay
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA5154013
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
513.68 | 5.95 | 5.95 |
520.69 | 5.41 | 5.41 |
494.71 | 5.25 | 5.25 |
549.73 | 5.85 | 5.85 |
544.72 | 5.88 | 5.88 |
573.75 | 5.40 | 5.40 |
415.61 | 4.21 | 4.21 |
554.15 | 6.67 | 6.67 |
483.73 | 5.69 | 5.69 |
534.73 | 5.46 | 5.46 |
504.14 | 6.03 | 6.03 |
519.64 | 5.90 | 5.90 |
586.78 | 4.16 | 4.16 |
541.76 | 5.17 | 5.17 |
508.74 | 5.64 | 5.64 |
570.79 | 4.41 | 4.41 |
501.72 | 5.91 | 5.91 |
509.67 | 4.31 | 4.31 |
576.83 | 4.17 | 4.17 |
576.83 | 4.17 | 4.17 |
454.64 | 4.41 | 4.41 |
497.67 | 3.18 | 3.18 |
601.81 | 6.03 | 6.03 |