Basic Information
ID: ALA5155250
Type: Binding
Description: Displacement of sapitinib-BODIPY tracer from C-terminal NanoLuc-fused full length wild type EGFR (unknown origin) transfected in HEK293T cells incubated for 2 hrs by NanoBRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293T
Target: Epidermal growth factor receptor erbB1(ALA203)
Document: ALA5154643
Displacement of sapitinib-BODIPY tracer from C-terminal NanoLuc-fused full length wild type EGFR (unknown origin) transfected in HEK293T cells incubated for 2 hrs by NanoBRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5155250
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 499.62 | 4.51 | 4.51 |
| 475.55 | 5.88 | 5.88 |
| 383.40 | 3.32 | 3.32 |
| 636.67 | 5.71 | 5.71 |
| 477.52 | 4.92 | 4.92 |
| 769.81 | 7.63 | 7.63 |
| 622.68 | 6.07 | 6.07 |