ID: ALA5156554
Type: Binding
Description: Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA5156554
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
386.46 | 3.78 | 3.78 |
450.43 | 3.80 | 3.80 |
534.61 | 6.97 | 6.97 |
448.45 | 3.52 | 3.52 |
435.46 | 3.47 | 3.47 |
476.51 | 4.79 | 4.79 |
424.41 | 4.08 | 4.08 |
447.47 | 3.81 | 3.81 |
436.44 | 3.52 | 3.52 |
464.50 | 4.16 | 4.16 |
464.45 | 3.73 | 3.73 |
421.43 | 3.01 | 3.01 |
420.44 | 3.73 | 3.73 |
422.42 | 3.13 | 3.13 |
462.48 | 4.49 | 4.49 |
519.53 | 4.28 | 4.28 |
437.43 | 2.29 | 2.29 |
434.43 | 3.75 | 3.75 |
434.47 | 3.99 | 3.99 |
449.44 | 3.04 | 3.04 |
436.44 | 3.43 | 3.43 |
448.45 | 3.93 | 3.93 |
506.53 | 4.38 | 4.38 |
450.47 | 3.77 | 3.77 |
512.54 | 5.01 | 5.01 |
435.46 | 2.88 | 2.88 |
461.50 | 4.37 | 4.37 |
450.43 | 3.64 | 3.64 |
440.86 | 4.60 | 4.60 |
474.41 | 4.96 | 4.96 |
533.56 | 4.85 | 4.85 |