Assay Report Card

Basic Information

ID: ALA5156583

Type: Binding

Description: Binding affinity to His6-tagged human BRDT bromodomain-2 (257 to 382 residues) expressed in Escherichia coli BL21 (DE3) assessed as increase in thermal stability by measuring change in melting temperature at 200 uM incubated for 30 mins by SYPRO orange dye based thermal shift assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
386.463.783.78
534.616.976.97
476.514.794.79
421.433.013.01
519.534.284.28
461.504.374.37