Basic Information
ID: ALA5158073
Type: Binding
Description: Inhibition of human recombinant NEK1 (1 to 505 residues) assessed as residual activity at 1 uM using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric scintillation counting assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5158073
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 344.44 | 2.07 | 2.07 |
| 356.45 | 2.17 | 2.17 |
| 407.50 | 3.11 | 3.11 |
| 416.50 | 3.03 | 3.03 |
| 281.32 | 1.95 | 1.95 |
| 331.40 | 2.15 | 2.15 |
| 372.49 | 2.85 | 2.85 |
| 423.49 | 2.82 | 2.82 |
| 331.40 | 1.84 | 1.84 |
| 407.50 | 3.11 | 3.11 |
| 386.48 | 1.84 | 1.84 |
| 359.41 | 2.07 | 2.07 |
| 317.37 | 1.50 | 1.50 |
| 421.48 | 3.20 | 3.20 |
| 423.49 | 2.82 | 2.82 |
| 446.53 | 3.59 | 3.59 |
| 345.42 | 2.28 | 2.28 |
| 446.53 | 3.59 | 3.59 |
| 384.51 | 2.99 | 2.99 |