Basic Information
ID: ALA5158663
Type: Binding
Description: Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate measured after 1 hr by HTRF assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5158663
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 280.37 | 5.03 | 5.03 |
| 362.43 | 4.98 | 4.98 |
| 377.39 | 3.54 | 3.54 |
| 302.38 | 4.96 | 4.96 |
| 405.45 | 4.19 | 4.19 |
| 321.42 | 3.57 | 3.57 |
| 352.38 | 5.55 | 5.55 |
| 268.36 | 4.88 | 4.88 |
| 442.97 | 5.14 | 5.14 |
| 282.39 | 5.27 | 5.27 |
| 303.37 | 4.36 | 4.36 |
| 320.37 | 5.10 | 5.10 |
| 401.47 | 3.28 | 3.28 |
| 359.40 | 3.40 | 3.40 |
| 316.40 | 5.27 | 5.27 |
| 316.40 | 5.52 | 5.52 |
| 370.37 | 5.98 | 5.98 |
| 321.42 | 3.53 | 3.53 |
| 369.47 | 4.17 | 4.17 |
| 341.41 | 3.26 | 3.26 |
| 369.47 | 3.91 | 3.91 |
| 338.36 | 5.24 | 5.24 |
| 356.43 | 3.00 | 3.00 |