Assay Report Card

Basic Information

ID: ALA5161277

Type: Binding

Description: Antagonist activity at human TRPV1 expressed in CHO cells assessed as low pH-induced Ca2+ influx at 10 uM incubated for 30 mins at pH 5 by FLIPR method

Organism: Homo sapiens

Cell type: CHO

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
429.244.264.26
418.505.875.87
391.546.306.30
400.515.735.73
391.546.306.30
394.465.095.09
397.485.335.33
418.505.875.87
401.895.975.97
385.445.465.46
377.515.805.80
367.455.325.32
408.485.405.40
417.466.206.20