Basic Information
ID: ALA5162524
Type: Binding
Description: Inhibition of C-terminal His6-tagged BRD4 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 hrs by HTRF assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5162524
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 457.00 | 5.53 | 5.53 |
| 491.56 | 5.06 | 5.06 |
| 630.76 | 6.88 | 6.88 |
| 594.64 | 6.22 | 6.22 |
| 623.67 | 6.46 | 6.46 |
| 610.64 | 5.90 | 5.90 |
| 540.55 | 5.33 | 5.33 |
| 554.58 | 5.58 | 5.58 |
| 580.61 | 6.29 | 6.29 |
| 529.61 | 7.09 | 7.09 |
| 636.67 | 6.43 | 6.43 |
| 622.69 | 6.84 | 6.84 |
| 634.73 | 6.76 | 6.76 |
| 564.61 | 6.91 | 6.91 |
| 642.65 | 6.42 | 6.42 |
| 575.61 | 6.75 | 6.75 |
| 527.60 | 6.84 | 6.84 |
| 599.70 | 7.62 | 7.62 |
| 515.59 | 6.53 | 6.53 |
| 602.63 | 7.12 | 7.12 |
| 651.73 | 7.24 | 7.24 |
| 596.61 | 5.67 | 5.67 |
| 557.62 | 6.47 | 6.47 |
| 547.55 | 6.02 | 6.02 |
| 588.61 | 6.87 | 6.87 |
| 637.70 | 6.85 | 6.85 |
| 571.65 | 6.86 | 6.86 |
| 638.69 | 6.67 | 6.67 |
| 568.60 | 6.14 | 6.14 |
| 526.56 | 5.46 | 5.46 |
| 644.79 | 7.13 | 7.13 |
| 624.66 | 6.29 | 6.29 |
| 536.56 | 6.30 | 6.30 |
| 574.58 | 6.48 | 6.48 |
| 616.74 | 6.62 | 6.62 |
| 569.68 | 8.01 | 8.01 |
| 600.62 | 6.87 | 6.87 |
| 594.64 | 6.68 | 6.68 |
| 541.62 | 7.23 | 7.23 |
| 555.65 | 7.62 | 7.62 |
| 638.69 | 6.68 | 6.68 |
| 566.59 | 5.90 | 5.90 |
| 648.73 | 6.02 | 6.02 |
| 526.52 | 5.02 | 5.02 |