Assay Report Card

Basic Information

ID: ALA5164356

Type: Functional

Description: Antagonist activity at human MC5R transfected in HEK293 cells co-transfected with GScAMP22F assessed as decrease in alpha-MSH induced cAMP level at 0.1 to 0.000001 M in presence of 500 nM alpha-MSH by split luciferase cAMP sensor dynamic assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1601.84
1561.82