Basic Information
ID: ALA5165903
Type: Binding
Description: Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system assessed as residual activity at 1 uM using ARTKQTARKSTGGKAPRKQLA as substrate measured after 30 mins in presence of ATP by ADP-Glo assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5165903
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 328.40 | 4.37 | 4.37 |
| 270.36 | 3.26 | 3.26 |
| 292.35 | 3.09 | 3.09 |
| 298.42 | 4.04 | 4.04 |
| 358.38 | 3.13 | 3.13 |
| 314.37 | 3.98 | 3.98 |
| 256.22 | 2.09 | 2.09 |
| 272.29 | 2.81 | 2.81 |
| 240.22 | 2.27 | 2.27 |
| 284.39 | 3.65 | 3.65 |
| 242.31 | 2.48 | 2.48 |
| 284.39 | 3.65 | 3.65 |
| 273.39 | 3.62 | 3.62 |
| 270.36 | 3.26 | 3.26 |
| 286.32 | 3.20 | 3.20 |
| 300.34 | 3.59 | 3.59 |
| 314.37 | 3.98 | 3.98 |
| 256.33 | 2.87 | 2.87 |
| 300.34 | 3.59 | 3.59 |
| 226.24 | 1.77 | 1.77 |