Basic Information
ID: ALA5165908
Type: Binding
Description: Inhibition of recombinant rat DYRK1A (1 to 499 residues ) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate measured after 30 mins in presence of ATP by ADP-Glo assay
Organism: Rattus norvegicus
Activity Charts
Bioactivity
Activity Types for Assay ALA5165908
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 270.36 | 3.26 | 3.26 |
| 292.35 | 3.09 | 3.09 |
| 256.22 | 2.09 | 2.09 |
| 272.29 | 2.81 | 2.81 |
| 240.22 | 2.27 | 2.27 |
| 284.39 | 3.65 | 3.65 |
| 242.31 | 2.48 | 2.48 |
| 270.36 | 3.26 | 3.26 |
| 286.32 | 3.20 | 3.20 |