Assay Report Card

Basic Information

ID: ALA5166186

Type: Binding

Description: Activation of human 20S proteosome at caspase-like site assessed as maximum fold change in substrate degradation using Z-LLE-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
381.885.935.93
353.876.156.15
381.885.935.93
492.987.987.98
368.856.056.05
338.865.735.73