Basic Information
ID: ALA5166774
Type: Binding
Description: Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation constant of SRC3 using FAM-labeled +H3N-KKENNALLRYLLDRDDPSD-CO2- peptide as substrate incubated overnight followed by substrate addition incubated for overnight by fluorescence polarization assay (Rvb = 7 microM)
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5166774
Kd
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 464.68 | 6.09 | 6.09 |
| 550.77 | 6.71 | 6.71 |
| 472.67 | 7.91 | 7.91 |