Assay Report Card

Basic Information

ID: ALA5166988

Type: Binding

Description: Binding affinity to CDK8 in human HCT-116 cells assessed as reduction in protease-induced CDK8 degradation at 1 to 4 uM treated for 6 hrs followed by protease treatment for 30 mins by western blot analysis

Organism: Homo sapiens

Cell type: HCT-116

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
414.513.613.61