Basic Information
ID: ALA5167481
Type: Functional
Description: Antagonist activity at human RXFP3 expressed in CHO-K1 cells assessed as forskolin-induced cAMP accumulation measured after 30 mins in presence of relaxin-3 by TR-FRET assay
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA5167481
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 507.47 | 4.80 | 4.80 |
| 482.54 | 3.85 | 3.85 |
| 445.52 | 4.17 | 4.17 |
| 466.54 | 5.01 | 5.01 |
| 470.50 | 4.84 | 4.84 |
| 452.51 | 4.70 | 4.70 |
| 469.50 | 3.79 | 3.79 |
| 458.54 | 4.76 | 4.76 |
| 458.54 | 4.76 | 4.76 |
| 453.50 | 4.09 | 4.09 |
| 453.50 | 4.09 | 4.09 |
| 438.49 | 4.70 | 4.70 |
| 457.47 | 3.92 | 3.92 |
| 452.51 | 4.70 | 4.70 |
| 470.50 | 4.84 | 4.84 |
| 518.37 | 4.55 | 4.55 |
| 2622.09 | ||
| 453.50 | 4.09 | 4.09 |
| 473.92 | 4.44 | 4.44 |
| 482.54 | 4.71 | 4.71 |
| 467.53 | 4.35 | 4.35 |
| 453.50 | 4.09 | 4.09 |
| 418.50 | 4.16 | 4.16 |
| 466.54 | 4.74 | 4.74 |
| 481.56 | 4.91 | 4.91 |
| 442.48 | 4.29 | 4.29 |
| 470.50 | 4.84 | 4.84 |
| 462.89 | 4.64 | 4.64 |
| 439.48 | 3.79 | 3.79 |
| 452.51 | 4.70 | 4.70 |
| 453.50 | 4.09 | 4.09 |