Assay Report Card

Basic Information

ID: ALA5216112

Type: Binding

Description: Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate incubated for 30 mins by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
163.180.500.50
214.230.800.80
174.202.232.23
248.342.282.28
229.313.023.02
281.330.560.56
253.351.101.10
261.672.462.46
221.281.721.72
262.28-1.30-1.30
221.251.321.32
243.231.211.21
235.312.682.68
305.192.732.73
266.332.352.35
209.230.970.97
199.212.532.53
194.20-1.48-1.48
264.312.272.27
269.763.223.22
239.301.201.20
201.191.251.25
310.401.541.54
198.272.402.40